Clinical Pharmacology Details


IVERMECTIN


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Indications & Dose:


Strongyloidiasis:


Adult and Child > 15 kg 


PO 3 mg (15-24 kg), 6mg (25-35 kg), 9mg (36-50kg), 12mg (51-65kg), 15mg (66-79 kg), 200ug/kg (>80kg)


Onchocerciasis:



PO 3 mg (15-24 kg), 6mg (25-35 kg), 9mg (36-50 kg), 12mg (51-65 kg), 15mg (66-79 kg), 150 ug/kg (>80kg)


Ascariasis:



PO 50-200 ug/kg


Enterobiasis:



PO 50-200 ug/kg


Trichuriasis:



PO 200ug/kg qd X 2 days


Scabies:



TOP 0.8% solution applied to entire body; PO 12mg

Contraindications:

Side Effects:

CNS: Dizziness, somnolence, tremor, vertigo


GI: Anorexia, constipation, diarrhea, increased transaminase levels, nausea 


HEME: Leukopenia


SKIN: Pruritus, rash, urticaria


MISC.: Fatigue 

Cautions:

Precautions:

 Rapid killing of microfilariae may induce systemic or ocular inflammatory response (Mazzotti reaction) 

Interaction:

Warnings:

Adverse Effects:

Lactations:

Pregnancy category C; excreted in breast milk in low concentrations 

Special Precautions:

Counselling:

Side Effects Or Adverse Reactions:

Patient And Carer Advice: