Clinical Pharmacology Details


PIPERAZINE CITRATE


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Indications & Dose:


Adults


Threadworm: 50-75mg piperazine base/kg body wt. daily for 7 days.


Ascariasis:



Single dose of 750mg piperazine hexahydrate for each year of age. Maximum of 4.5mg.


Children 50-75mg/kg/dose on two consecutive nights for Ascariasis for oxyuriasis 25-50mg/kg/day for 7 days. 

Contraindications:

Side Effects:

Nausea, vomiting, colic, diarrhea, allergy like urticaria, bronchospasm and rare reports of Stevens.  Johnson syndrome and angioedema, rarely dizziness, muscular incoordination, drowsiness, confusion and clonic contractions in patients with neurological & renal abnormalities. 

Cautions:

Renal impairment  (avoid if  severe), liver disease, neurological disease, epilepsy, pregnancy

Precautions:

Neurological disturbances.  Safety not established.


Breast-feeding: Safety not established.


Old age: May be used. 

Interaction:

Drugs


Pyrantal pamoate: Antagonism. 

Warnings:

Adverse Effects:

Lactations:

Special Precautions:

Counselling:

Side Effects Or Adverse Reactions:

Patient And Carer Advice: