Clinical Pharmacology Details


Dexamethasone


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Indications & Dose:

Suppression of inflammatory and allergic disorders



Adult: 0.5–10 mg daily


Mild croup



Child: 150 micrograms/kg for 1 dose


Severe croup (or mild croup that might cause complications)



Child: Initially 150 micrograms/kg for 1 dose, to be given before transfer to hospital, then (by mouth or byintravenous injection) 150 micrograms/kg, then (bymouth or by intravenous injection) 150 micrograms/kgafter 12 hours if required


Congenital adrenal hyperplasia (under expert supervision)



Adult: Consult specialist for advice on dosing


Corticosteroid responsive conditions



Adult: Consult specialist for advice on dosing


Overnight dexamethasone suppression test



Adult: 1 mg for 1 dose, to be given at night


Adjunctive treatment of bacterial meningitis (starting before or with first dose of antibacterial)



Adult: 8.3 mg every 6 hours for 4 days


Symptom control of anorexia (in palliative care)


Adult: 2–4 mg daily


Obstruction due to tumour (dysphagia in palliative care)


Adult: 8 mg daily


Bronchospasm or partial obstruction (dyspnoea in palliative care)


Adult: 4–8 mg daily


Nausea and vomiting (adjunct in palliative care)



Adult: 8–16 mg daily


Headaches due to raised intracranial pressure (in palliative care)


Adult: 16 mg daily for 4–5 days, then reduced to 4–6 mg daily, reduce dose if possible. To be given before 6pm to reduce the risk of insomnia


Pain due to nerve compression (in palliative care)


Adult: 8 mg daily


Cerebral oedema associated with malignancy



Adult: 0.5–10 mg daily


Cerebral oedema



Adult: Initially 8–16 mg for 1 dose, then (by intramuscular injection or by intravenous injection) 5 mg every 6 hours until adequate response achieved then taper-off gradually, use the 3.8 mg/ mL injection preparation for this dose


Cerebral oedema associated with malignancy



Adult: Initially 8.3 mg for 1 dose, then (by intramuscular injection) 3.3 mg every 6 hours as required for 2–4 days, subsequently, reduce dose gradually and stop over 5–7 days, use the 3.3 mg/ mL injection preparation for this dose


• Shock:


IV 1-6 mg/kg or 40 mg q26h (phosphate)


• Prophylaxis during premature labor (to prevent infant respiratory distress due to immature lungs):


6 mg q 12h x 4 doses


Intralesional:


0.8-1.6 mg (acetate)


• Intra-articular and soft tissue:


4-16 mg q l-3 wk (acetate); large joints 2-4 mg (phosphate); small joints 0.8-1 mg (phosphate); bursae 23 mg (phosphate); tendon sheaths 0.41 mg (phosphate); soft tissue infiltration 2-6 mg (phosphate); ganglia 1-2 mg (phosphate) 

Contraindications:

Systemic fungal infections; (ophth): acute superficialherpes simplex keratitis and other viral diseases of the cornea and conjunctiva; fungal diseases of ocular structures; ocular TB; following uncomplicated removal of a superficial corneal foreign body. Pregnancy. 

Side Effects:

CNS: Depression, headache, moodchanges, seizures,vertigo
CV: CHF,hypertension, tachycardia,thromboernbolism, thrombophlebitis
EENT: Blurred vision, cataracts, dryness, epistaxis, increased intraocular pressure, localized infections of nose and pharynx with C. albicans, nasal irritation, nasal septum perforation, rebound congestion, sneezing, sore throat, stinging (nasal); cataracts, decreased acuity, glaucoma exacerbation, increased intraocular pressure, increased probability of corneal infection, optic nerve damage, poor corneal wound healing, stinging, transient burning (ophth)
GI: Abdominal distention, diarrhea, GI hemorrhage,increased appetite, nausea, pancreatitis
GU: Hypercalciuria
METAB: Cushingoid state, decreased glucose tolerance, decreased t4, growth suppression in children, HPA suppression, hyperglycemia
MS: Aseptic necrosis of femoral and humeraI heads, fractures, myopathy, osteoporosis, weakness
SKIN: Acne, bruising, ecchymosis, petechiae, poor wound healing, striae, suppression of skin test reactions, thin fragile skin 

Cautions:

Precautions:

Psychosis, cerebral malaria, elderly, AIDS, latent tuberculosis or amebiasis (reactivation of disease), diabetes mellitus, glaucoma, osteoporosis, ulcerative colitis (intestinal perforation), CHF, myasthenia gravis, renal disease, esophagitis, peptic ulcer, hypertension; (ophth): infections of the eye, glaucoma.


Breast-feeding: Use with caution
Old age: Use with caution. 

Interaction:

Drugs


Aminoglutethamide: Enhanced elimination of corticosteroids; marked reduction in corticosteroid response; increased clearance of dexamethasone; doubling of dose may be necessary


Antidiabetics: Increased blood glucose


Barbiturates, carbamazepine:Reduced serum concentrations of corticosteroids; increased clearance of dexamethasone


Cholestyramine, colestipol: Possible reduced absorption of corticosteroids


Cyclosporirne: Possible increased concentration of both drugs, seizures


Erythromycin, troleandomycin, clarithromycin, ketoconazole: Possible enhanced steroid effect


Estrogens, oral contraceptives:Enhanced effects of corticosteroids Isoniazid: Reduced plasma concentrations of isoniazid


IUDs: Inhibition of inflammation may decrease contraceptive effect


NSAIDs: Increased risk GI ulceration


Rifampin: Reduced therapeutic effect of corticosteroids; may reduce hepatic clearance of prednisone


Salicylates: Subtherapeutic salicylate concentrations possible


 

Warnings:

Adverse Effects:

Lactations:

Special Precautions:

Counselling:

Side Effects Or Adverse Reactions:

Patient And Carer Advice: