Clinical Pharmacology Details


Oestradiol VALERATE


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Indications & Dose:

HRT for menopausal symptoms due to oestrogen deficiency, postmeno pausal osteoporosis and clinical conditions requiring natural oestradiol (E2) replacement including primary ovarian failure, hyperandrogenism in females.


DOSE


Adult: One tab once a day for 21 days.


Child: Not recommended.

Contraindications:

Pregnancy carcinoma of endometrium, carcinoma of breast, hepatic damage, thromboembolic disorder, thrombosis, endometriosis, vaginal bleeding of unknown cause.


 

Side Effects:

Nausea, vomiting, weight gain, breast tenderness & enlargement, jaundice, rashes ,withdrawl bleeding. Pruritus, exan-thema, thrombophlebitis, local skin irritation. 

Cautions:

Hypertension, myocardial or renal disease, asthma, varicose vein, epilepsy, fibromyometa. 

Precautions:

Epilepsy, migraine, cardiac failure, hypertension, diabetes mellitus, fibrocystic disease of breast, hepatic and renal dysfunction.


BREAST-FEEDING: Use with caution. 

Interaction:

Drugs


Same as ethinyl estradiol

Warnings:

Adverse Effects:

Lactations:

Special Precautions:

Counselling:

Side Effects Or Adverse Reactions:

Patient And Carer Advice: